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Composition:
Each tablet contains:
Metronidazole: 400 mg
Description: Metronidaziole is
an Nitroimidazole derivative effective against
anaerobic Protozoa like T. vaginalis, E.histolytica,
G.lamblia and non sporing anaerobic Gram negative
bacilli such as bacterioides.It is an effective
systemic Trichomonocide.It is rapidly absorbed
through small bowel. Food does not effect its
absorption. Metronidazole diffuses in all tissues
and achieves high concentrations in CSF, bile,
bone and abcess and hence causes Lethal effect
on Sensitive bacteria at therapeutic doses . It
enters the microorganism by diffusion,
Its Nitro group is reduced to intermediate compound
which causes cytotoxicity probably by damaging
DNA .Its selectively high activity against anaerobic
bacteria has suggested interference with electron
transport from NADPH or other reduced substance.
Metronidazole is almost completely absorbed from
small intestine and is widely distributed in the
body attaining therapeutic concentration in Vaginal
secretions, Saliva, semen, CSF.
Indications:
*Used in chronic Amoebiasis.
*Used in diarrhoea and dysentery caused by Bacteria
or Protozoa.
*It is also used in treatment of Trichomonas Vaginitis,
Anaerobic infections
(after colorectal or pelvic surgery, appendectomy,
Osteomyelitis, Brain or lung abcess )
* Used in ulcerative gingivitis, bacterial Enterites,
food poisioning, giardiasis.
Contraindications:
*Intolerance to Alcohol.
*Primaquine sensitivity, infants below one month.
* Blood dyscrasis and Neurological disorders.
Pregnancy: First trimester of
Pregnancy contraindicated
Lactation: Contraindicated.
Dosage: 1 Tablet three times
a Day.
Presentation: 20x10 tablets in
a Multicarton.
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